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CAS No.: 1642303-38-5
Synonyms: ITI214 Phosphate
ITI-214 is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and ion channels, exhibits potent PDE1 inhibitory activity (Ki = 58 pM).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03257046 | Parkinson Disease | Phase 1 Phase 2 | Recruiting | August 2018 | United States, Georgia ... more >> Atlanta Center for Medical Research Recruiting Atlanta, Georgia, United States, 30331 United States, North Carolina Duke Early Phase Research Unit Recruiting Durham, North Carolina, United States, 27708 Collapse << |
NCT03387215 | Heart Failure, Systolic | Phase 1 Phase 2 | Recruiting | December 2019 | United States, Maryland ... more >> Johns Hopkins University Recruiting Baltimore, Maryland, United States, 21287 Principal Investigator: Nisha Gilotra, MD United States, North Carolina Duke Clinical Research Institute Recruiting Durham, North Carolina, United States, 27710 Collapse << |
NCT03489772 | Healthy Volunteers | Phase 1 | Recruiting | June 2019 | United States, Oklahoma ... more >> Laureate Institute for Brain Research, Inc. Recruiting Tulsa, Oklahoma, United States, 74136 Principal Investigator: Sahib S Khalsa, MD, PhD Collapse << |
实验方案
技术信息
CAS号 | 1642303-38-5 | 储存条件 |
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分子式 | C29H29FN7O5P | 运输 | 蓝冰 | |||
分子量 | 605.56 | 别名 | ITI214 Phosphate | |||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03257046 | Parkinson Disease | Phase 1 Phase 2 | Recruiting | August 2018 | United States, Georgia ... more >> Atlanta Center for Medical Research Recruiting Atlanta, Georgia, United States, 30331 United States, North Carolina Duke Early Phase Research Unit Recruiting Durham, North Carolina, United States, 27708 Collapse << |
NCT03387215 | Heart Failure, Systolic | Phase 1 Phase 2 | Recruiting | December 2019 | United States, Maryland ... more >> Johns Hopkins University Recruiting Baltimore, Maryland, United States, 21287 Principal Investigator: Nisha Gilotra, MD United States, North Carolina Duke Clinical Research Institute Recruiting Durham, North Carolina, United States, 27710 Collapse << |
NCT03489772 | Healthy Volunteers | Phase 1 | Recruiting | June 2019 | United States, Oklahoma ... more >> Laureate Institute for Brain Research, Inc. Recruiting Tulsa, Oklahoma, United States, 74136 Principal Investigator: Sahib S Khalsa, MD, PhD Collapse << |
NCT01900522 | Schizophrenia | Phase 1 | Terminated(Business Decision; ... more >>No Safety or Efficacy Concerns) Collapse << | - | United States, California ... more >> Glendale, California, United States United States, New York New York, New York, United States Collapse << |
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